Synthesis of 1-triazolyl-4-trimethylsilyl-2-butanol and 1-triazolyl-5-trimethylsilyl-2-pentanol derivatives and an investigation of their fungicidal activities.

نویسندگان

  • Hiroyuki Itoh
  • Rieko Yoneda
  • Junzo Tobitsuka
  • Hiroshi Ohta
  • Yukiyoshi Takahi
  • Mikio Tsuda
  • Hideo Takeshiba
چکیده

A new series of azole derivatives of 1-triazolyl-4-trimethylsilyl-2-butanol and 1-triazolyl-5-trimethylsilyl-2-pentanol were synthesized and evaluated for fungicidal activities against rice blast, sheath blight, and powdery mildew on barley. The derivatives of 2,4-difluorobenzene exhibited high antifungal activities when applied by spray, but exhibited no fungicidal activity by submerged application.

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عنوان ژورنال:
  • Chemical & pharmaceutical bulletin

دوره 51 9  شماره 

صفحات  -

تاریخ انتشار 2003